SCHEMBL19937816

SCHEMBL19937816

CC1(Cn2ccc(-c3cnc(N)c(C(F)(F)F)c3)n2)CC1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 18/20 0.52
TNF P01375 1/20 0.44
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19937608 0.81 MAP3K12 (0.52) MAP3K12TNFPIK3CA
SCHEMBL19937665 0.79 MAP3K12 (0.52) MAP3K12TNF
SCHEMBL19937631 0.77 MAP3K12 (0.54) MAP3K12TNF
SCHEMBL19937793 0.74 MAP3K12 (0.52) MAP3K12TNFPIK3CA
SCHEMBL19937616 0.73 MAP3K12 (0.57) MAP3K12TNFPIK3CA
SCHEMBL19937784 0.73 MAP3K12 (0.39) MAP3K12PIK3CA
SCHEMBL19937787 0.72 MAP3K12 (0.54) MAP3K12TNF
SCHEMBL19937642 0.71 MAP3K12 (0.55) MAP3K12TNF
SCHEMBL19937751 0.71 MAP3K12 (0.53) MAP3K12TNF
SCHEMBL18403198 0.69 MAP3K12 (1.00) MAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945938-B1 3-SUBSTITUTED PYRAZOLES AND USE AS DLK INHIBITORS HOFFMANN LA ROCHE (CH) 2018-03-07 EP disclosed