SCHEMBL19944820

SCHEMBL19944820

CCCNC1C=C(CO)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.35
DRD3 P35462 5/20 0.35
DRD4 P21917 2/20 0.35
CES2 O00748 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP1B1 Q16678 1/20 0.34
ALDH1A1 P00352 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR1A P08908 2/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19944817 0.70 DRD3 (0.42) DRD2DRD3DRD4HTR1A
SCHEMBL2908570 0.69 CES2 (0.36) CES2ALOX15CYP1B1ALDH1A1
SCHEMBL5888258 0.67
SCHEMBL16119131 0.66
SCHEMBL9062785 0.66
SCHEMBL1532221 0.64 DRD3 (0.36) DRD3CES2ALOX15CYP1B1ALDH1A1
SCHEMBL1071437 0.60 CNR1 (0.39) DRD3CES2ALOX15CYP1B1ALDH1A1
SCHEMBL27480307 0.59 EPHX2 (0.32)
SCHEMBL7962273 0.58
SCHEMBL19433041 0.57 CES2 (0.34) CES2ALOX15CYP1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018044136-A1 NOVEL COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT FOR PREVENTING OR TREATING DISEASES ASSOCIATED WITH POLY(ADP-RIBOSE) POLYMERASE-1 (PARP-1) 충남대학교 산학협력단 2018-03-08 WO disclosed