SCHEMBL1994570

SCHEMBL1994570

CSCc1csc(C(F)(F)F)n1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.34
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ATM Q13315 1/20 0.32
SLC6A3 Q01959 1/20 0.31
IDH1 O75874 1/20 0.31
HRH1 P35367 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9262966 0.79 MCHR1 (0.34) MCHR1GAAIDH1HRH1
SCHEMBL17263328 0.76 CCR4 (0.40) MCHR1IDH1HRH1
SCHEMBL12607354 0.75 IDH1 (0.33) MCHR1IDH1
SCHEMBL127293 0.75 IDH1 (0.33) MCHR1IDH1
SCHEMBL1999685 0.75 SRC (0.35) MCHR1IDH1
SCHEMBL5437866 0.75 IDH1 (0.36) MCHR1IDH1
SCHEMBL1569158 0.75 IDH1 (0.33) MCHR1ALDH1A1IDH1
SCHEMBL9045575 0.75 GFER (0.42) MCHR1GAAKMT2AALDH1A1IDH1
SCHEMBL5329328 0.75 IDH1 (0.33) MCHR1IDH1
SCHEMBL1912967 0.74 IDH1 (0.33) MCHR1IDH1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2338885-B1 Insecticidal N-Substituted (2-Substituted-1,3-Thiazol) Alkyl Sulfoximines DOW AGROSCIENCES LLC (US) 2012-10-31 EP disclosed
EP-2057135-B1 INSECTICIDAL N-SUBSTITUTED (2- SUBSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES DOW AGROSCIENCES LLC (US) 2012-06-13 EP disclosed
US-8183270-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES, LLC (US) 2012-05-22 US disclosed
US-8183270-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES, LLC (US) 2012-05-22 US disclosed
EP-2338885-A1 Insecticidal N-Substituted (2-Substituted-1,3-Thiazol) Alkyl Sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338883-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338884-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
EP-2338884-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines Dow AgroSciences LLC (US) 2011-06-29 EP disclosed
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES CORTEVA AGRISCIENCE LLC 2011-03-10 US disclosed
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES CORTEVA AGRISCIENCE LLC 2011-03-10 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
US-7863303-B2 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2011-01-04 US disclosed
EP-2057135-A1 INSECTICIDAL N-SUBSTITUTED (2- SUDSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES Dow AgroSciences LLC (US) 2009-05-13 EP disclosed
WO-2008027539-A1 INSECTICIDAL N-SUBSTITUTED (2- SUDSTITUTED-1,3-THIAZOL) ALKYL SULFOXIMINES DOW AGROSCIENCES LLC (US) 2008-03-06 WO disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines DOW AGROSCIENCES LLC (US) 2008-03-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080058394-A1 Insecticidal N-substituted (2-substituted-1,3-thiazol)alkyl sulfoximines TST, NIT2, MSL1 MCHR1 2202/4885GAA 4482/4885MEN1 2936/4885
US-20110060018-A1 INSECTICIDAL N-SUBSTITUTED (2-SUBSTITUTED-1,3-THIAZOL)ALKYL SULFOXIMINES TST, NIT2, MSL1 MCHR1 2202/4885GAA 4482/4885MEN1 2936/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.