SCHEMBL19953017

SCHEMBL19953017

Fc1ccc(F)c(-c2cncn2-c2ccc(OC(F)(F)F)cc2)c1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
HTR6 P50406 2/20 0.35
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HSP90AA1 P07900 7/20 0.34
HSP90AB1 P08238 7/20 0.34
PPARD Q03181 2/20 0.34
PPARA Q07869 2/20 0.34
RXRA P19793 2/20 0.34
GRIN1 Q05586 2/20 0.34
GRIN2B Q13224 2/20 0.34
HTR2A P28223 1/20 0.33
SCN5A Q14524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953054 0.88 IDO1 (0.39) PTGS2HTR6HTR1AHTR7POLB
SCHEMBL19953047 0.81 HSP90AA1 (0.45) HSP90AA1HSP90AB1
SCHEMBL19953125 0.74 CYP11B2 (0.37) HTR6HTR1AHTR7HSP90AA1HSP90AB1
SCHEMBL19953046 0.71 HSP90AA1 (0.41) HTR6HTR1AHTR7HSP90AA1HSP90AB1
SCHEMBL19953001 0.71 HSP90AA1 (0.42) PTGS2HTR6HTR1AHTR7HSP90AA1
SCHEMBL6290646 0.69 PTGS2 (0.64) PTGS2
SCHEMBL1071938 0.69 HSP90AA1 (0.50) HTR6HSP90AA1HSP90AB1HTR2A
SCHEMBL19953094 0.69 HSP90AA1 (0.44) PTGS2HSP90AA1HSP90AB1
SCHEMBL19953061 0.69 HSP90AA1 (0.51) HSP90AA1HSP90AB1
SCHEMBL27933810 0.69 NPY5R (0.48) MAOAMAOBSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed