SCHEMBL19953048

SCHEMBL19953048

Cc1ncn(-c2ccc(Cl)cc2)c1-c1c(F)cccc1F

nearest known ligand 0.79

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.42
PTGS1 P23219 1/20 0.42
RAB9A P51151 1/20 0.41
GRM1 Q13255 1/20 0.40
CYP11B2 P19099 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953042 0.88 PTGS2 (0.43) PTGS2RAB9ACYP11B2
SCHEMBL19953052 0.86 PTGS2 (0.41) PTGS2PTGS1RAB9ACYP11B2
SCHEMBL19953173 0.85 PTGS2 (0.50) PTGS2PTGS1RAB9A
SCHEMBL1074163 0.82 PTGS2 (0.42) PTGS2PTGS1RAB9AGRM1CYP11B2
SCHEMBL19967375 0.78 PTGS2 (0.67) PTGS2PTGS1CYP11B2
SCHEMBL1082336 0.73 PDE2A (0.40) RAB9A
SCHEMBL1072687 0.73 PDE2A (0.40) RAB9AGRM1
SCHEMBL19953091 0.73 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL23507084 0.72 MKNK1 (0.47) PTGS2RAB9AGRM1CYP11B2
SCHEMBL19214262 0.72 ALDH1A1 (0.50) PTGS2RAB9AGRM1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed