SCHEMBL19953243

SCHEMBL19953243

COCCCOc1cc2c(nc1OC)-c1cc(=O)c(C(=O)O)cn1C(C(C)(C)C)C2

nearest known ligand 0.77

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2B6 P20813 1/20 0.77
TENT4A Q5XG87 1/20 0.77
TENT4B Q8NDF8 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20876569 1.00 CYP2B6 (0.77) CYP2B6TENT4ATENT4B
SCHEMBL19966858 0.91 CYP2B6 (0.64) CYP2B6TENT4ATENT4B
SCHEMBL29579831 0.91 CYP2B6 (0.64) CYP2B6TENT4ATENT4B
SCHEMBL20876573 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL20876562 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL20876563 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL20876593 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL20876574 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL20876594 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B
SCHEMBL30137678 0.90 CYP2B6 (0.63) CYP2B6TENT4ATENT4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200255428-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-08-13 US claimed
EP-3692040-A1 CHEMICAL COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-08-12 EP claimed
WO-2019069293-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-11 WO claimed
US-20250066361-A1 5,6,7,7a-Tetrahydrocyclopenta[f]pyrido[1,2-h][1,7] naphthyridin-11(4bH)-one Compounds and Methods of use Use (as amended) GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2025-02-27 US disclosed
US-12221444-B2 5,6,7,7a-tetrahydrocyclopenta[f]pyrido[1,2-h][1,7]naphthyridin-11(4bH)-one compounds and methods of use GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2025-02-11 US disclosed
EP-4180431-A1 CHEMICAL COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2023-05-17 EP disclosed
EP-3692040-B1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE IP DEV LTD (GB) 2022-12-28 EP disclosed
US-20220144834-A1 Chemical Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2022-05-12 US disclosed
US-20210330678-A1 PAPD5 INHIBITORS AND METHODS OF USE THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-10-28 US disclosed
US-20200255428-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-08-13 US disclosed
EP-3692040-A1 CHEMICAL COMPOUNDS GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-08-12 EP disclosed
WO-2019069293-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-11 WO disclosed
WO-2018047109-A1 POLYCYCLIC PYRIDONE COMPOUNDS AS ANTIVIRALS NOVARTIS AG (CH) 2018-03-15 WO disclosed
WO-2018047109-A1 POLYCYCLIC PYRIDONE COMPOUNDS AS ANTIVIRALS NOVARTIS AG (CH) 2018-03-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12221444-B2 5,6,7,7a-tetrahydrocyclopenta[f]pyrido[1,2-h][1,7]naphthyridin-11(4bH)-one compounds and methods of use HAVCR2, HBS1L, HBG1 CYP2B6 65/4885TENT4A 936/4885TENT4B 558/4885
US-20210330678-A1 PAPD5 INHIBITORS AND METHODS OF USE THEREOF PARP15, PAPSS1, PGA5 CYP2B6 3451/4885TENT4A 154/4885TENT4B 109/4885
US-20250066361-A1 5,6,7,7a-Tetrahydrocyclopenta[f]pyrido[1,2-h][1,7] naphthyridin-11(4bH)-one Compounds and Methods of use Use (as amended) HAVCR2, HMBS, HBS1L CYP2B6 19/4885TENT4A 1040/4885TENT4B 746/4885
US-20220144834-A1 Chemical Compounds HAVCR2, HBS1L, HLA-B CYP2B6 254/4885TENT4A 2212/4885TENT4B 1797/4885
US-20200255428-A1 CHEMICAL COMPOUNDS HAVCR2, HBS1L, HLA-B CYP2B6 254/4885TENT4A 2212/4885TENT4B 1797/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.