SCHEMBL19953390

SCHEMBL19953390

NCc1cc(=O)c2ccccc2s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 5/20 0.56
CYP2A6 P11509 4/20 0.56
ASIC3 Q9UHC3 1/20 0.56
ALDH1A1 P00352 4/20 0.55
ALOX15 P16050 2/20 0.55
MAPK1 P28482 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GPR3 P46089 1/20 0.41
MAPK3 P27361 1/20 0.41
MAP2K1 Q02750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1193947 0.81 ALDH1A1 (0.59) CYP2A6ALDH1A1ALOX15MAPK1MAPT
SCHEMBL11785606 0.79 ALDH1A1 (0.60) LOXL2ALDH1A1ALOX15MAPK1MAPT
SCHEMBL19953210 0.77 CYP2A6 (0.46) LOXL2CYP2A6ASIC3HPGD
SCHEMBL26752820 0.73 ALDH1A1 (0.49) ALDH1A1ALOX15MAPK1MAPTHPGD
SCHEMBL240588 0.72 CYP2A6 (1.00) LOXL2CYP2A6ASIC3AGXT
SCHEMBL1194406 0.71 ALDH1A1 (1.00) ALDH1A1ALOX15MAPK1MAPTHPGD
SCHEMBL7777304 0.71 ALDH1A1 (0.60) ALDH1A1ALOX15MAPK1MAPTHPGD
Hydrochloric Acid SCHEMBL6941951 0.71 CYP2A6 (0.96) LOXL2CYP2A6ASIC3AGXT
SCHEMBL466086 0.71 ALDH1A1 (1.00) ALDH1A1ALOX15MAPK1MAPTHPGD
Iodide SCHEMBL30536902 0.71 CYP2A6 (0.96) LOXL2CYP2A6ASIC3AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048928-A1 CHEMICAL PROBES OF LYSYL OXIDASE-LIKE 2 AND USES THEREOF PHARMAKEA, INC. (US) 2018-03-15 WO disclosed
WO-2018048930-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2018-03-15 WO disclosed
WO-2018048930-A1 LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2018-03-15 WO disclosed