SCHEMBL19953485

SCHEMBL19953485

CN1CCC(C(=O)NC2Cc3ccccc3C2)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.44
FABP5 Q01469 1/20 0.43
EPHX2 P34913 1/20 0.42
HRH3 Q9Y5N1 4/20 0.42
HTR6 P50406 1/20 0.42
MTNR1A P48039 3/20 0.42
MTNR1B P49286 3/20 0.42
GRM7 Q14831 2/20 0.40
TRPV1 Q8NER1 1/20 0.39
P2RX4 Q99571 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
IDO1 P14902 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960927 0.81 KCNQ2 (0.44) KCNQ2FABP5EPHX2HRH3HTR6
SCHEMBL19953533 0.80 FABP5 (0.43) FABP5EPHX2HRH3HTR6MTNR1A
SCHEMBL19953489 0.80 FABP5 (0.43) FABP5EPHX2HRH3HTR6MTNR1A
SCHEMBL19953584 0.80 FABP5 (0.43) FABP5EPHX2HRH3HTR6MTNR1A
SCHEMBL28279788 0.77 KDM4C (0.43) KCNQ2HTR6MTNR1AMTNR1BTRPV1
SCHEMBL30899464 0.76 KDM4C (0.44) HTR6MTNR1AMTNR1BTRPV1KDM4C
SCHEMBL16250257 0.76 KDM4C (0.44) HTR6MTNR1AMTNR1BTRPV1KDM4C
SCHEMBL19127981 0.75 KDM4C (0.42) TRPV1KDM4CNPC1RAB9A
SCHEMBL19953514 0.75 OPRM1 (0.43) KCNQ2FABP5EPHX2HRH3MTNR1A
SCHEMBL20778981 0.75 KDM4C (0.41) HTR6MTNR1AMTNR1BTRPV1KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO claimed
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed