SCHEMBL1995440

SCHEMBL1995440

CCc1ccc(O)cc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.57
CA1 P00915 4/20 0.57
CA2 P00918 4/20 0.57
CA7 P43166 4/20 0.57
CA9 Q16790 4/20 0.57
CA14 Q9ULX7 4/20 0.57
ALOX5 P09917 1/20 0.57
PTGS2 P35354 1/20 0.57
ALDH1A1 P00352 4/20 0.52
TSHR P16473 1/20 0.52
HSD17B10 Q99714 2/20 0.50
MYC P01106 1/20 0.49
PTPN1 P18031 1/20 0.49
HSP90AB1 P08238 1/20 0.46
EGFR P00533 2/20 0.45
LCK P06239 2/20 0.45
HSD17B1 P14061 1/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140476 0.86 CA12 (0.52) CA12CA1CA2CA7CA9
SCHEMBL14674137 0.85 CA12 (0.59) CA12CA1CA2CA7CA9
SCHEMBL17926251 0.83 TYR (0.61) CA12CA1CA2CA7CA9
SCHEMBL28126806 0.83 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL39010 0.83 CA12 (0.57) CA12CA1CA2CA7CA9
SCHEMBL15782801 0.83 HSD17B1 (0.58) CA12CA1CA2CA7CA9
SCHEMBL9959316 0.82 CA2 (0.55) CA12CA1CA2CA7CA9
SCHEMBL27658957 0.82 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL27517848 0.82 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL3873135 0.82 CA12 (0.55) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016008862-A1 SUBSTITUTED VINYL AND ALKYNYL CYANOCYCLOALKANOLS AND VINYL AND ALKYNYL CYANOHETEROCYCLOALKANOLS AS ACTIVE AGENTS AGAINST ABIOTIC PLANT STRESS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-01-21 WO disclosed
CN-102361857-B Can be used as the ring-type benzimidizole derivatives of antidiabetic MERCK SHARP & DOHME CORP. (US) 2015-09-16 CN disclosed
WO-2012139891-A1 SUBSTITUTED VINYL AND ALKINYL CYCLOHEXENOLS AS ACTIVE AGENTS AGAINST ABIOTIC STRESS IN PLANTS BAYER CROPSCIENCE AG (DE) 2012-10-18 WO disclosed
US-7960417-B2 Such as 1-(2,2-dimethylpropyl)-4-propyl-5-{4-[4-(1H-tetrazol-5-yl)phenoxy]butoxy}-1H-indole; neurological and psychiatric disorders MERCK SHARP & DOHME CORP. (US) 2011-06-14 US disclosed
CN-101941964-A Has the Chemokine Receptors bonded heterogeneous ring compound that promotes effect ANORMED INC 2011-01-12 CN disclosed
CN-1826310-B Novel aminobenzophenone compounds LEO PHARMA AS 2010-07-21 CN disclosed
CN-101426786-A Benzazole potentiators of metabotropic glutamate receptors MERCK & CO INC (US) 2009-05-06 CN disclosed
US-20080176904-A1 Benzazole Potentiators of Metabotropic Glutatmate Receptors MERCK SHARP & DOHME CORP. 2008-07-24 US disclosed
EP-1855670-A2 BENZAZOLE POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS Merck & Co., Inc. (US) 2007-11-21 EP disclosed
CN-1282636-C Vitamin D analogues GALDERMA RES & DEV (FR) 2006-11-01 CN disclosed
WO-2006091496-A2 BENZAZOLE POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERCK & CO., INC. (US) 2006-08-31 WO disclosed
CN-1826310-A Novel aminobenzophenone compounds LEO PHARMA AS (DK) 2006-08-30 CN disclosed
CN-1332711-A Vitamin D analogues GALDERMA RES & DEV (FR) 2002-01-23 CN disclosed
US-3985797-A Hydroxylation of aromatic compounds UOP INC. (US) 1976-10-12 US disclosed
US-3985796-A Hydroxylation of aromatic compounds UOP INC. (US) 1976-10-12 US disclosed
US-3931295-A Hydroxylation of aromatic compounds UNIVERSAL OIL PRODUCTS COMPANY (US) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176904-A1 Benzazole Potentiators of Metabotropic Glutatmate Receptors GRM2, GRM3, GRIK2 CA12 4211/4885CA1 2573/4885CA2 863/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.