SCHEMBL19954680

SCHEMBL19954680

O=C1/C(=C/c2ccc(Cl)c(Cl)c2)CN(C(=O)[C@@H](Cc2ccccc2)NC2CCCC2)C/C1=C\c1ccc(Cl)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 2/20 0.44
HSP90AA1 P07900 1/20 0.44
CARM1 Q86X55 5/20 0.42
NOS2 P35228 1/20 0.41
PSMB5 P28074 1/20 0.41
PTGS2 P35354 1/20 0.39
BCHE P06276 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
P4HB P07237 1/20 0.38
FPR2 P25090 1/20 0.38
GPR183 P32249 1/20 0.38
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
MDM2 Q00987 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21303814 0.89 PAX8 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL24253327 0.87 PSMB5 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL24253325 0.87 PSMB5 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL23334290 0.87 PSMB5 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL21303829 0.87 PAX8 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL22221603 0.87 PAX8 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL17693759 0.87 PAX8 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL21303828 0.86 PAX8 (0.46) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL22851690 0.85 CARM1 (0.41) PAX8HSP90AA1CARM1NOS2PSMB5
SCHEMBL25179856 0.85 PAX8 (0.45) PAX8HSP90AA1CARM1NOS2PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9913834-B2 Bis-benzylidine piperidone proteasome inhibitor with anticancer activity THE JOHNS HOPKINS UNIVERSITY (US) 2018-03-13 US disclosed