SCHEMBL19954967

SCHEMBL19954967

C[C@@]1(c2nc3ccccc3[nH]2)CCCN1C(=O)I

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.51
HCRTR2 O43614 20/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19954979 0.83 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL665171 0.79 PARP1 (0.58) HCRTR1HCRTR2
SCHEMBL665626 0.76 PARP1 (0.60) HCRTR1HCRTR2
SCHEMBL665107 0.76 PARP1 (0.47) HCRTR1HCRTR2
SCHEMBL665994 0.74 PARP1 (0.58) HCRTR1HCRTR2
SCHEMBL10522199 0.74 HRH4 (0.39) HCRTR1HCRTR2
SCHEMBL15559527 0.74 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL16798917 0.72 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL16778810 0.71 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL4965847 0.71 ALDH1A1 (0.43) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9914721-B2 Use of benzimidazole-proline derivatives IDORSIA PHARMACEUTICALS LTD (CH) 2018-03-13 US disclosed