SCHEMBL19955442

SCHEMBL19955442

CC(=O)Nc1cccc(C(=O)C(C)C)c1C(C)=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.46
POLB P06746 2/20 0.46
CYP2C19 P33261 2/20 0.46
KDM4E B2RXH2 3/20 0.46
HSD17B10 Q99714 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.39
MAPK1 P28482 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ALOX15 P16050 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17399834 0.84 CYP2C19 (0.53) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL19955438 0.84 CYP2C19 (0.44) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL22299425 0.83 CYP2C19 (0.61) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL27634334 0.81 POLB (0.54) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL24113861 0.75 THRB (0.39) KDM4EHSD17B10ALDH1A1HPGDNPC1
SCHEMBL9377084 0.75 POLB (0.54) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL11519154 0.74 CYP2C19 (0.53) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL4732713 0.74 KDM4E (0.54) POLBCYP2C19KDM4EHSD17B10KMT2A
SCHEMBL11593694 0.73 POLB (0.56) MAOAPOLBCYP2C19KDM4EHSD17B10
SCHEMBL30346643 0.73 POLB (0.56) MAOAPOLBCYP2C19KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2663549-B1 PHENETHYLSULFONE ISOINDOLINE DERIVATIVES AS INHIBITORS OF PDE 4 AND/OR CYTOKINES CELGENE CORP (US) 2018-03-14 EP disclosed