SCHEMBL4732713

SCHEMBL4732713

COC(=O)c1cccc(NC(=O)C(C)C)c1C(C)=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.54
ALDH1A1 P00352 4/20 0.54
LMNA P02545 2/20 0.51
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
HPGD P15428 2/20 0.48
GAA P10253 1/20 0.48
MDM4 O15151 2/20 0.47
TP53 P04637 2/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 2/20 0.45
CETP P11597 1/20 0.45
POLB P06746 1/20 0.45
ATM Q13315 1/20 0.45
BDKRB1 P46663 1/20 0.44
HSD17B10 Q99714 3/20 0.43
USP2 O75604 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5928724 0.83 TSHR (0.68) KDM4EALDH1A1LMNATSHRTDP1
SCHEMBL8893471 0.82 KDM4E (0.50) KDM4EALDH1A1LMNATSHRTDP1
SCHEMBL4732717 0.79 ALDH1A1 (0.49) KDM4EALDH1A1LMNATSHRTDP1
SCHEMBL31590548 0.76 LMNA (0.53) KDM4EALDH1A1LMNATSHRHPGD
SCHEMBL4026343 0.76 LMNA (0.53) KDM4EALDH1A1LMNATSHRHPGD
SCHEMBL8908317 0.74 POLB (0.50) KDM4EALDH1A1LMNATSHRHPGD
SCHEMBL16281636 0.74 MDM4 (0.51) KDM4EALDH1A1LMNAMDM4TP53
SCHEMBL19955442 0.74 MAOA (0.46) KDM4EALDH1A1LMNATSHRHPGD
SCHEMBL6164745 0.73 KDM4E (0.51) KDM4EALDH1A1LMNATSHRTDP1
SCHEMBL1663385 0.72 CA12 (0.59) KDM4EALDH1A1TSHRTDP1MDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008054454-A2 NITROGEN-CONTAINING HETEROCYCLE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF AS ANTIVIRAL AGENTS TRANSTECH PHARMA, INC. (US) 2008-05-08 WO disclosed