SCHEMBL19955676

SCHEMBL19955676

COC(=O)Cc1c(C)c2c(c(C)c1-c1cc(F)c3c(c1C)CCCO3)CNC2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.37
KLKB1 P03952 5/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18944215 0.91 NR1I2 (0.36) NR1I2KLKB1ALDH1A1
SCHEMBL19955759 0.88 NR1I2 (0.38) NR1I2MEN1ALDH1A1GAAMAPT
SCHEMBL18929663 0.86 NR1I2 (0.35) NR1I2MEN1ALDH1A1GAAMAPT
SCHEMBL19955789 0.85 NR1I2 (0.37) NR1I2MAPT
SCHEMBL19955514 0.85 NR1I2 (0.38) NR1I2MAPT
SCHEMBL18664243 0.83 NR1I2 (0.36) NR1I2MEN1ALDH1A1GAAMAPT
SCHEMBL19955743 0.80 NR1I2 (0.36) NR1I2MEN1ALDH1A1MAPTKMT2A
SCHEMBL18928959 0.80 NR1I2 (0.33) NR1I2
SCHEMBL19955744 0.79 NR1I2 (0.33) NR1I2
SCHEMBL19955611 0.77 NR1I2 (0.41) NR1I2MEN1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166925-B1 ISOINDOLINE DERIVATIVES FOR USE IN THE TREATMENT OF A VIRAL INFECTION VIIV HEALTHCARE UK LTD (GB) 2018-03-14 EP disclosed