SCHEMBL18664243

SCHEMBL18664243

CCOC(=O)Cc1c(C)c2c(c(C)c1-c1cc(F)c3c(c1C)CCCO3)CCNCC2

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.36
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 2/20 0.31
CASP1 P29466 2/20 0.31
CASP7 P55210 2/20 0.31
HSD17B10 Q99714 2/20 0.31
GLA P06280 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
HTT P42858 1/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18944215 0.92 NR1I2 (0.36) NR1I2KDM4EALDH1A1HSD17B10HPGD
SCHEMBL18663914 0.86 NR1I2 (0.37) NR1I2
SCHEMBL18944148 0.85 NR1I2 (0.38) NR1I2
SCHEMBL19955676 0.83 NR1I2 (0.37) NR1I2ALDH1A1MAPTGAASMN1; SMN2
SCHEMBL18546248 0.81 NR1I2 (0.40) NR1I2KDM4EALDH1A1LMNAHSD17B10
SCHEMBL18928972 0.80 NR1I2 (0.33) NR1I2
SCHEMBL18928302 0.80 LMNA (0.40) NR1I2KDM4EALDH1A1LMNAMAPT
SCHEMBL18928959 0.80 NR1I2 (0.33) NR1I2
SCHEMBL18929005 0.79 NR1I2 (0.36) NR1I2MAPTKMT2A
SCHEMBL18928142 0.79 HTR4 (0.33) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017046707-A1 BENZOAZEPINE DERIVATIVES VIIV HEALTHCARE UK LIMITED (GB) 2017-03-23 WO disclosed