SCHEMBL19955759

SCHEMBL19955759

COC(=O)Cc1c(C)c2c(c(C)c1-c1cc(F)c3c(c1C)CCCO3)CN(C)C2

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.38
MAPT P10636 2/20 0.34
THRB P10828 1/20 0.34
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19955514 0.90 NR1I2 (0.38) NR1I2MAPTTHRB
SCHEMBL19955789 0.90 NR1I2 (0.37) NR1I2MAPTTHRB
SCHEMBL19955591 0.89 NR1I2 (0.39) NR1I2
SCHEMBL19955676 0.88 NR1I2 (0.37) NR1I2MAPTMEN1ALDH1A1GAA
SCHEMBL18929725 0.87 NR1I2 (0.36) NR1I2MAPTTHRB
SCHEMBL19955743 0.84 NR1I2 (0.36) NR1I2MAPTTHRBMEN1ALDH1A1
SCHEMBL19955627 0.84 NR1I2 (0.35) NR1I2
SCHEMBL19955744 0.83 NR1I2 (0.33) NR1I2
SCHEMBL18944148 0.82 NR1I2 (0.38) NR1I2
SCHEMBL19955611 0.82 NR1I2 (0.41) NR1I2MAPTTHRBMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166925-B1 ISOINDOLINE DERIVATIVES FOR USE IN THE TREATMENT OF A VIRAL INFECTION VIIV HEALTHCARE UK LTD (GB) 2018-03-14 EP disclosed