SCHEMBL199582

SCHEMBL199582

O=Cc1c(I)ccnc1F

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NAPRT Q6XQN6 1/20 0.31
ERN1 O75460 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29836949 1.00 CCR1 (0.32) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL31492595 0.81 MEN1 (0.38) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL846251 0.81 MEN1 (0.38) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL18297654 0.78 ERN1 (0.35) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL25195292 0.77 ALDH1A1 (0.48) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL30356708 0.77 ALDH1A1 (0.48) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL26457513 0.77 CCR1 (0.33) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL4322219 0.75 ERN1 (0.38) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL31146149 0.75 NR4A2 (0.32) CCR1CCR5CCR8MEN1ALDH1A1
SCHEMBL5006077 0.75 ERN1 (0.41) CCR1CCR5CCR8MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 258 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637467-B2 Inhibitor of BTK and mutants thereof NEWAVE PHARMACEUTICAL INC. (US) 2026-05-26 US disclosed
US-12441743-B2 Spiro aromatic ring compound and use thereof ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2025-10-14 US disclosed
US-20250214970-A1 PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS XENON PHARMACEUTICALS INC. (CA) 2025-07-03 US disclosed
US-20250059189-A1 PYRIDINE DERIVATIVES AND THEIR USE AS SODIUM CHANNEL ACTIVATORS XENON PHARMACEUTICALS INC. (CA) 2025-02-20 US disclosed
EP-4055019-B1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING BTK VIA UBIQUITIN PROTEOSOME PATHWAY NURIX THERAPEUTICS INC (US) 2025-01-22 EP disclosed
US-12054486-B2 Pyridine derivatives and their use as sodium channel activators XENON PHARMACEUTICALS INC. (CA) 2024-08-06 US disclosed
EP-4405347-A1 PYRIDINE DERIVATIVES AND THEIR USE AS SODIUM CHANNEL ACTIVATORS Xenon Pharmaceuticals Inc. (CA) 2024-07-31 EP disclosed
CN-118271240-A Protein site-specific labeling probe and labeling method based on reversible Michael addition triggering o-group participating reaction 南开大学 2024-07-02 CN disclosed
CN-118284602-A Pyridine derivatives as sodium channel activators and uses thereof 泽农医药公司 2024-07-02 CN disclosed
US-20240116949-A1 SPIRO AROMATIC RING COMPOUND AND USE THEREOF ETERN BIOPHARMA SHANGHAI CO LTD (CN) 2024-04-11 US disclosed
WO-2005070891-A2 COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2005-08-04 WO disclosed
CN-1552712-A New camptothecin analogue compounds, a process for their preparation and pharmaceutical compositions containing them ɪά��ʵ���� 2004-12-08 CN disclosed
CN-1158282-C Camptothecin analogue compounds, preparation method thereof and pharmaceutical compositions containing same ɪά��ʵ���� 2004-07-21 CN disclosed
US-6699876-B2 FOR CANCER THERAPY LES LABORATOIRES SERVIER (FR) 2004-03-02 US disclosed
US-20030105109-A1 For cancer therapy LES LABORATOIRES SERVIER (FR) 2003-06-05 US disclosed
US-6509345-B2 For therapy of cancerous diseases LES LABORATOIRES SERVIER (FR) 2003-01-21 US disclosed
EP-1101765-B1 Camptothecin analogues, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2002-08-14 EP disclosed
US-20020077325-A1 New camptothecin analogue compounds LAVIELLE GILBERT (FR) 2002-06-20 US disclosed
CN-1301701-A Camptothecin analogue compounds, preparation method thereof and pharmaceutical compositions containing same ADIR (FR) 2001-07-04 CN disclosed
EP-1101765-A2 Camptothecin analogues, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-05-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030105109-A1 For cancer therapy OXER1, OXGR1, CBR1 CCR1 18/4885CCR5 226/4885CCR8 134/4885
US-20020077325-A1 New camptothecin analogue compounds OXER1, CBR3, CBR1 CCR1 29/4885CCR5 98/4885CCR8 147/4885
US-20240116949-A1 SPIRO AROMATIC RING COMPOUND AND USE THEREOF PTPN1, PTPN11, PTPN5 CCR1 687/4885CCR5 976/4885CCR8 1040/4885
US-12441743-B2 Spiro aromatic ring compound and use thereof PTPN1, PTPN11, PTPN5 CCR1 687/4885CCR5 976/4885CCR8 1040/4885
US-12637467-B2 Inhibitor of BTK and mutants thereof BTK, CNKSR1, SYK CCR1 431/4885CCR5 579/4885CCR8 1286/4885
US-20250214970-A1 PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS SCN1A, SCN3A, SCN2A CCR1 4186/4885CCR5 4815/4885CCR8 3885/4885
US-12054486-B2 Pyridine derivatives and their use as sodium channel activators SCN1A, SCN1B, CACNA1A CCR1 3587/4885CCR5 4635/4885CCR8 3945/4885
US-20250059189-A1 PYRIDINE DERIVATIVES AND THEIR USE AS SODIUM CHANNEL ACTIVATORS SCN1A, SCN1B, CACNA1A CCR1 3759/4885CCR5 4640/4885CCR8 3938/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.