SCHEMBL19959608

SCHEMBL19959608

CCSC(CC(C)=O)c1cccc(C#N)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.42
FFAR1 O14842 1/20 0.41
GRM4 Q14833 1/20 0.39
GSK3B P49841 2/20 0.38
GPR139 Q6DWJ6 1/20 0.38
S1PR1 P21453 1/20 0.37
KCNA5 P22460 2/20 0.37
ADRA1D P25100 3/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA1A P35348 1/20 0.37
CNR1 P21554 3/20 0.36
CNR2 P34972 3/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19959671 0.83 MAPT (0.43) GSK3BMEN1ALDH1A1MAPTKMT2A
SCHEMBL8895206 0.78 PDPK1 (0.43) MEN1ALDH1A1MAPTKMT2A
SCHEMBL23468143 0.75 TNF (0.40) TNFFFAR1GRM4GSK3BGPR139
SCHEMBL3937793 0.70 FFAR1 (0.56) TNFFFAR1GRM4GPR139KCNA5
SCHEMBL14762502 0.70 GRM4 (0.48) TNFFFAR1GRM4GSK3BGPR139
SCHEMBL1043636 0.69 PDCD1 (0.51) TNFFFAR1GRM4GSK3BGPR139
Benzonitrile SCHEMBL7358669 0.69 FFAR1 (0.49) TNFFFAR1GRM4GPR139MAPT
SCHEMBL200244 0.68 ERCC1 (0.52) FFAR1GSK3BCNR1
SCHEMBL9646909 0.68 LMNA (0.52) TNFFFAR1GRM4GSK3BGPR139
SCHEMBL30860058 0.68 ERCC1 (0.52) FFAR1GSK3BCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049296-A1 HETEROARYL INHIBITORS OF PAD4 PADLOCK THERAPEUTICS, INC. (US) 2018-03-15 WO disclosed