SCHEMBL19959671

SCHEMBL19959671

CCSC(CC(C)=O)c1ccc(C#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HTT P42858 2/20 0.40
ALDH1A1 P00352 1/20 0.38
CYP2A6 P11509 1/20 0.37
F2R P25116 1/20 0.36
GSK3B P49841 2/20 0.36
SLC6A3 Q01959 1/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
MMP12 P39900 1/20 0.34
MMP13 P45452 1/20 0.34
MGLL Q99685 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19959608 0.83 TNF (0.42) MAPTALDH1A1GSK3BMEN1KMT2A
SCHEMBL8895206 0.79 PDPK1 (0.43) MAPTKDM4EALDH1A1SLC6A3MEN1
SCHEMBL28509173 0.76 MAPT (0.48) MAPTKDM4EGAAL3MBTL1HTT
SCHEMBL28509175 0.76 MAPT (0.48) MAPTKDM4EGAAL3MBTL1HTT
SCHEMBL6370632 0.76 FFAR1 (0.50) MAPTKDM4EGAAL3MBTL1HTT
SCHEMBL23876831 0.72 MAPT (0.40) MAPTKDM4EGAAL3MBTL1HTT
SCHEMBL19959669 0.72 P2RX7 (0.35) MAPTKDM4EMEN1KMT2ATSHR
SCHEMBL19939827 0.69 ALDH1A1 (0.57) MAPTKDM4EGAAL3MBTL1HTT
SCHEMBL18029866 0.68 MAOA (0.50) MAPTKDM4EGAAL3MBTL1ALDH1A1
SCHEMBL2649430 0.68 CTBP2 (0.56) MAPTHTTALDH1A1CYP2A6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049296-A1 HETEROARYL INHIBITORS OF PAD4 PADLOCK THERAPEUTICS, INC. (US) 2018-03-15 WO disclosed