SCHEMBL19960929

SCHEMBL19960929

COC1c2ccccc2CC1NC(=O)C1c2ccccc2CC(=O)N1CC1CCOCC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.49
KCNH2 Q12809 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
TSHR P16473 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.33
RECQL P46063 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPT P10636 1/20 0.32
GAA P10253 1/20 0.32
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
PYGL P06737 1/20 0.31
NAMPT P43490 1/20 0.31
BRD4 O60885 1/20 0.31
F2 P00734 1/20 0.31
HTR4 Q13639 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960687 0.94 GRM7 (0.55) GRM7TSHRALDH1A1LMNARECQL
SCHEMBL20165965 0.88 GRM7 (0.46) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL20165963 0.88 GRM7 (0.46) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL20165964 0.88 GRM7 (0.46) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19960841 0.86 GRM7 (0.49) GRM7KCNH2SCN5ASCN9ALMNA
SCHEMBL19960865 0.86 GRM7 (0.51) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19960866 0.86 GRM7 (0.51) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19960834 0.84 GRM7 (0.45) GRM7KCNH2SCN5ASCN9ALMNA
SCHEMBL19953497 0.83 GRM7 (0.55) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL21542219 0.82 GRM7 (0.51) GRM7TSHRALDH1A1LMNARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed