SCHEMBL19953497

SCHEMBL19953497

O=C(NC1Cc2ccccc2C1)C1c2ccccc2CC(=O)N1CC1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.55
TSHR P16473 3/20 0.39
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MCHR1 Q99705 1/20 0.37
ALDH1A1 P00352 2/20 0.36
KCNH2 Q12809 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
BCL2 P10415 1/20 0.36
TP53 P04637 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
CCR1 P32246 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19953513 0.92 GRM7 (0.62) GRM7TSHRMAPTGAANPSR1
SCHEMBL19953654 0.92 GRM7 (0.62) GRM7TSHRMAPTGAANPSR1
SCHEMBL19960865 0.85 GRM7 (0.51) GRM7TSHRMAPTGAANPSR1
SCHEMBL19960866 0.85 GRM7 (0.51) GRM7TSHRMAPTGAANPSR1
SCHEMBL19960841 0.84 GRM7 (0.49) GRM7KCNH2SCN5ASCN9A
SCHEMBL19960661 0.83 GRM7 (0.53) GRM7
SCHEMBL19953548 0.83 GRM7 (0.53) GRM7
SCHEMBL19960929 0.83 GRM7 (0.49) GRM7TSHRMAPTGAANPSR1
SCHEMBL19953664 0.81 HRH3 (0.46) GRM7TSHRMAPTGAAALDH1A1
SCHEMBL19953510 0.81 HRH3 (0.46) GRM7TSHRMAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO claimed
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed