SCHEMBL19960865

SCHEMBL19960865

N[C@H]1c2ccccc2C[C@@H]1NC(=O)C1c2ccccc2CC(=O)N1CC1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 1/20 0.51
KCNH2 Q12809 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
TSHR P16473 2/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.32
NAMPT P43490 3/20 0.32
NPSR1 Q6W5P4 1/20 0.31
MCHR1 Q99705 1/20 0.31
F2 P00734 1/20 0.31
TACR2 P21452 1/20 0.31
GAA P10253 1/20 0.31
CNR2 P34972 3/20 0.31
CNR1 P21554 2/20 0.31
HTT P42858 1/20 0.31
ALDH1A1 P00352 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19960866 1.00 GRM7 (0.51) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19953650 0.93 GRM7 (0.57) GRM7TSHRMAPTLMNANPSR1
SCHEMBL19960690 0.93 GRM7 (0.57) GRM7TSHRMAPTLMNANPSR1
SCHEMBL19960841 0.87 GRM7 (0.49) GRM7KCNH2SCN5ASCN9ALMNA
SCHEMBL19960929 0.86 GRM7 (0.49) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19953497 0.85 GRM7 (0.55) GRM7KCNH2SCN5ASCN9ATSHR
SCHEMBL19960834 0.83 GRM7 (0.45) GRM7KCNH2SCN5ASCN9ALMNA
SCHEMBL19960507 0.82 GRM7 (0.58) GRM7TSHRMAPTLMNAGAA
SCHEMBL19953548 0.79 GRM7 (0.53) GRM7NAMPTTACR2CNR2CNR1
SCHEMBL19960661 0.79 GRM7 (0.53) GRM7NAMPTTACR2CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047983-A1 INDANE DERIVATIVES USEFUL AS MODULATORS OF MGLUR7 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-15 WO disclosed