SCHEMBL19964868

SCHEMBL19964868

CCOC(=O)c1cc2c(C)ccn2c(Cl)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.45
ALDH1A1 P00352 4/20 0.45
GLA P06280 3/20 0.45
GAA P10253 2/20 0.45
HPGD P15428 2/20 0.45
BAZ2B Q9UIF8 1/20 0.45
BAZ2A Q9UIF9 1/20 0.45
TSHR P16473 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAPK1 P28482 2/20 0.42
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
HSD17B10 Q99714 2/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19964719 0.86 KDM4E (0.49) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL19964974 0.82 KDM4E (0.44) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL21113451 0.75 KDM4E (0.40) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL19964720 0.75 EZH2 (0.41) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL19964970 0.71 HTT (0.42) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL19964413 0.69 KDM4E (0.48) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL7104912 0.69 KDM4E (0.51) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL21342092 0.69 KDM4E (0.47) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL17331626 0.68 ALDH1A1 (0.56) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL1444977 0.68 MAPK1 (0.46) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045971-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发有限公司 2018-03-15 WO disclosed