SCHEMBL19966646

SCHEMBL19966646

CCN1CCN(C(=O)c2ccc(Nc3ncc(F)c(-c4cc(F)c5cnn(C(C)C)c5c4)n3)nc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 17/20 0.65
CDK4 P11802 2/20 0.65
CCND3 P30281 2/20 0.65
CCND1 P24385 13/20 0.63
DYRK2 Q92630 3/20 0.62
PIM1 P11309 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19966302 0.90 CDK6 (0.66) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966573 0.87 CDK6 (0.64) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966649 0.85 CDK6 (0.63) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966544 0.85 CDK6 (0.71) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL17477168 0.84 CDK6 (0.75) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL17489238 0.82 CDK6 (0.74) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19209837 0.81 CDK6 (0.69) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966382 0.81 CDK6 (0.71) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966325 0.80 CDK6 (0.61) CDK6CDK4CCND3CCND1DYRK2
SCHEMBL19966456 0.80 CDK6 (0.56) CDK6CDK4CCND3CCND1DYRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018045957-A1 CDK4/6 INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 江苏豪森药业集团有限公司 2018-03-15 WO disclosed