SCHEMBL19967247

SCHEMBL19967247

C/C=N\C(C)=C(/C)c1c(F)cccc1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.40
CES1 P23141 3/20 0.40
TDP1 Q9NUW8 2/20 0.37
ERN1 O75460 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 3/20 0.33
TRPA1 O75762 1/20 0.33
LMNA P02545 2/20 0.32
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MEN1 O00255 1/20 0.31
KRAS P01116 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19967292 0.82 CES2 (0.42) CES2CES1TDP1KMT2ATRPA1
SCHEMBL19967289 0.71 TDP1 (0.40) CES2CES1TDP1ERN1POLB
SCHEMBL19967276 0.70 CES2 (0.46) CES2CES1TDP1ERN1POLB
SCHEMBL1990301 0.68 CES2 (0.55) CES2CES1TDP1ERN1POLB
SCHEMBL19102224 0.65 CES2 (0.64) CES2CES1TDP1ERN1POLB
SCHEMBL7924194 0.64 CES2 (0.50) CES2CES1TDP1ERN1POLB
SCHEMBL167447 0.64 CES2 (0.64) CES2CES1TDP1POLBKMT2A
SCHEMBL17055823 0.64 GAA (0.45) CES2CES1POLBKMT2AALDH1A1
SCHEMBL13458195 0.63 CES2 (0.39) CES2CES1TDP1ERN1KMT2A
Iodide SCHEMBL6190800 0.63 CES2 (0.48) CES2CES1TDP1ERN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed