SCHEMBL19967313

SCHEMBL19967313

Cc1ccc(F)c(-c2c(C)nc(C)n2-c2ccc(Cl)cc2)c1F

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GRM1 Q13255 3/20 0.36
PIK3CA P42336 1/20 0.36
GRM5 P41594 4/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1076197 0.92 POLB (0.38) POLBKDM4EGRM1PIK3CAGRM5
SCHEMBL19953205 0.89 POLB (0.36) POLBKDM4EGRM1PIK3CAGRM5
SCHEMBL1072687 0.86 PDE2A (0.40) POLBKDM4EGRM1PIK3CAGRM5
SCHEMBL1073294 0.82 PIK3CA (0.41) POLBKDM4EGRM1PIK3CAGRM5
SCHEMBL1075463 0.80 POLB (0.41) POLBKDM4EGRM1PIK3CAGRM5
SCHEMBL1075285 0.80 POLB (0.35) POLBKDM4EPIK3CAMEN1NPC1
SCHEMBL19953050 0.78 POLB (0.33) POLBKDM4EGRM5MEN1NPC1
SCHEMBL19953097 0.78 POLB (0.33) POLBKDM4EGRM5MEN1NPC1
SCHEMBL1073747 0.77 SMN1; SMN2 (0.41) POLBKDM4EPIK3CAGAA
SCHEMBL1073238 0.75 GRM5 (0.37) POLBPIK3CAGRM5NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018048969-A1 MULTI-TARGETED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-03-15 WO disclosed