SCHEMBL1073238

SCHEMBL1073238

COc1ccc(F)c(-c2c(C)nc(C)n2-c2ccc(F)cc2)c1F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.37
CYP2C9 P11712 2/20 0.36
GPBAR1 Q8TDU6 2/20 0.36
PIK3CA P42336 2/20 0.35
POLB P06746 1/20 0.34
BRD9 Q9H8M2 1/20 0.34
GRM8 O00222 1/20 0.34
CYP1A2 P05177 1/20 0.34
TACR1 P25103 1/20 0.34
GRM7 Q14831 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
USP2 O75604 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 2/20 0.33
KCNH2 Q12809 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MTOR P42345 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1224856 0.88 GRM5 (0.36) GRM5CYP2C9PIK3CAPOLBMAPT
SCHEMBL1225604 0.88 GPBAR1 (0.35) CYP2C9GPBAR1GRM8CYP1A2TACR1
SCHEMBL1073760 0.81 POLB (0.36) CYP2C9POLB
SCHEMBL1075218 0.80 HSP90AA1 (0.35) CYP2C9BRD9NPC1RAB9AMAPK1
SCHEMBL1074066 0.80 ALDH1A1 (0.34) CYP2C9GRM8CYP1A2TACR1GRM7
SCHEMBL1076510 0.79 PIK3CA (0.43) GRM5GPBAR1PIK3CAPOLBGRM8
SCHEMBL1073274 0.79 ALDH1A1 (0.37) CYP2C9GPBAR1NPC1RAB9AMAPK1
SCHEMBL1075665 0.79 PTGS2 (0.34) GPBAR1MAPT
SCHEMBL1076197 0.77 POLB (0.38) GRM5PIK3CAPOLB
SCHEMBL1075200 0.77 ALDH1A1 (0.36) GPBAR1MAPK1MAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056463-A2 FUNGICIDAL MIXTURES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-05-12 WO disclosed
US-20110045101-A1 FUNGICIDAL SUBSTITUTED AZOLES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2011-02-24 US disclosed
EP-2274284-A2 FUNGICIDAL SUBSTITUTED AZOLES E. I. Du Pont de Nemours and Company (US) 2011-01-19 EP disclosed
WO-2009137538-A2 FUNGICIDAL SUBSTITUTED AZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-11-12 WO disclosed
WO-2009137651-A2 FUNGICIDAL SUBSTITUTED AZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-11-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110045101-A1 FUNGICIDAL SUBSTITUTED AZOLES CBR3, NOX3, CBR1 GRM5 2940/4885CYP2C9 33/4885GPBAR1 3153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.