SCHEMBL19969375

SCHEMBL19969375

CCCc1cccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)OC)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.57
CTSK P43235 9/20 0.52
CTSS P25774 8/20 0.52
CTSB P07858 4/20 0.52
CTSL P07711 2/20 0.51
ACE P12821 1/20 0.50
POLB P06746 1/20 0.47
EPHX2 P34913 1/20 0.46
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32676816 0.90 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL2352344 0.85 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL2352336 0.85 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL30765043 0.85 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL6491302 0.85 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL29543144 0.85 KLK5 (0.59) KLK5CTSKCTSSCTSBCTSL
SCHEMBL2346583 0.84 CTSS (0.69) KLK5CTSKCTSSCTSBCTSL
SCHEMBL21946642 0.84 CTSS (0.69) KLK5CTSKCTSSCTSBCTSL
SCHEMBL6680700 0.84 KLK5 (0.61) KLK5CTSKCTSSCTSBCTSL
SCHEMBL4729306 0.84 KLK5 (0.58) KLK5CTSKCTSSCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018047139-A1 COMPOUNDS AS MODULATORS OF TIGIT SIGNALLING PATHWAY AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-15 WO disclosed