SCHEMBL19970520

SCHEMBL19970520

C#CCCCCOC[C@@H]1COC2(C=C(C(=O)O)C(S(=O)(=O)Cc3ccc(F)cc3Cl)CC2)O1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
TLR4 O00206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20111188 0.91 TLR4 (0.39) ALDH1A1GAATLR4
SCHEMBL19970532 0.85
SCHEMBL19970509 0.84 ALDH1A1 (0.35) ALDH1A1GAATLR4
SCHEMBL19970530 0.78 RORC (0.40) ALDH1A1GAA
SCHEMBL19970513 0.77 RORC (0.36) ALDH1A1GAA
SCHEMBL19970494 0.76 ALDH1A1 (0.34) ALDH1A1GAATLR4
SCHEMBL19970499 0.76 KMT2A (0.37) ALDH1A1GAATLR4
SCHEMBL19970495 0.76 CYP2D6 (0.34) ALDH1A1GAATLR4
SCHEMBL19970535 0.76 ALDH1A1 (0.37) ALDH1A1GAA
SCHEMBL19970497 0.76 ALDH1A1 (0.37) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180118708-A1 CYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-05-03 US disclosed
EP-3296296-A1 CYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2018-03-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180118708-A1 CYCLIC COMPOUND TLR4, TLR3, TLR9 ALDH1A1 973/4885GAA 4730/4885TLR4 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.