SCHEMBL19973163

SCHEMBL19973163

CC(C)(C)[Si](C)(C)OCCc1ccc2ncc(Br)n2c1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DUT P33316 2/20 0.32
PIK3CA P42336 1/20 0.30
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19973167 0.74 KEAP1 (0.50) DUT
SCHEMBL3458584 0.74 CYP11B1 (0.35) DUT
SCHEMBL19950913 0.73 SCN10A (0.33) PIK3CAMTOR
SCHEMBL408605 0.73 TAAR1 (0.40) DUT
SCHEMBL31132717 0.71 PIK3CA (0.39) PIK3CAMTOR
SCHEMBL19950877 0.70 SCN10A (0.30)
SCHEMBL9701756 0.70 DUT (0.36) DUT
SCHEMBL5871377 0.70 MEN1 (0.42) DUT
SCHEMBL17428939 0.69 KMT2A (0.41) DUT
SCHEMBL12002859 0.69 DUT (0.40) DUT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512833-A1 HETEROARYL CARBOXAMIDE COMPOUNDS AS INHIBITORS OF RIPK2 Boehringer Ingelheim International GmbH (DE) 2019-07-24 EP disclosed
WO-2018052772-A1 HETEROARYL CARBOXAMIDE COMPOUNDS AS INHIBITORS OF RIPK2 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-03-22 WO disclosed