SCHEMBL19974414

SCHEMBL19974414

COc1nc(Cl)nc2c1ncn2[C@@H]1O[C@H](C(O)CC(C)(OC)OC)[C@H]2OC(C)(C)OC[C@]21C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.34
HRH2 P25021 1/20 0.32
HTR5A P47898 1/20 0.32
ADORA3 P0DMS8 7/20 0.32
ADORA1 P30542 7/20 0.32
ADORA2B P29275 4/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22683313 0.81 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19974599 0.74 ADORA1 (0.40) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19978975 0.71 ADORA2A (0.41) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19974410 0.69 ADORA2A (0.64) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL6838477 0.65 ADORA2A (0.74) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19978907 0.64 ADORA1 (0.38) ADORA2AHRH2HTR5AADORA3ADORA1
SCHEMBL19975005 0.64 ADORA2A (0.46) ADORA2AADORA3
SCHEMBL27087637 0.64 LMNA (0.45) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19974564 0.64 ADORA2A (0.58) ADORA2AADORA3ADORA1ADORA2BALOX15
SCHEMBL19974415 0.64 ADORA2A (0.47) ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512860-A1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB Pharma Inc. (CA) 2019-07-24 EP disclosed
WO-2018049534-A1 NUCLEOSIDE AND NUCLEOTIDE ANALOGUES BEARING A QUATERNARY ALL-CARBON STEREOGENIC CENTER AT THE 2' POSITION AND METHODS OF USE AS A CARDIOPROTECTIVE AGENT LCB PHARMA INC. (CA) 2018-03-22 WO disclosed