SCHEMBL19974983

SCHEMBL19974983

NCc1noc([C@H]2CCCN2C(=O)OC(=O)C(F)(F)F)n1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.42
DPP8 Q6V1X1 5/20 0.42
DPP9 Q86TI2 5/20 0.42
DPP7 Q9UHL4 5/20 0.42
GRM5 P41594 9/20 0.39
HCRTR1 O43613 4/20 0.38
HCRTR2 O43614 4/20 0.38
PREP P48147 3/20 0.38
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL19974982 0.83 DPP4 (0.43) DPP4DPP8DPP9DPP7GRM5
Trifluoroacetic Acid SCHEMBL19974984 0.83 DPP4 (0.43) DPP4DPP8DPP9DPP7GRM5
SCHEMBL19979747 0.78 DPP4 (0.40) DPP4DPP8DPP9DPP7GRM5
SCHEMBL15175334 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL16933907 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL16934066 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL16934064 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL16933905 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL15175333 0.69 ALDH1A1 (0.55) ALDH1A1
SCHEMBL30147174 0.68 TSHR (0.49) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053302-A1 MACROCYCLIC COMPOUNDS FOR THE INHIBITION OF INDOLEAMINE-2,3-DIOXYGENASE ACTIVITY AND USE THEREOF ENSEMBLE THERAPEUTICS CORPORATION (US) 2018-03-22 WO disclosed