SCHEMBL19977052

SCHEMBL19977052

CC(NC(=O)c1ccccc1Br)C(=O)Nc1cccc2c1OCCO2

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.47
MAPT P10636 3/20 0.43
F2R P25116 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CTNNB1 P35222 1/20 0.38
WNT3A P56704 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19977128 0.91 F2R (0.45) MRGPRX1MAPTF2RALDH1A1LMNA
SCHEMBL19976912 0.88 MRGPRX1 (0.48) MRGPRX1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL19976937 0.87 TP53 (0.52) MRGPRX1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL19976991 0.87 MRGPRX1 (0.47) MRGPRX1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL19976896 0.84 SMN1; SMN2 (0.47) MRGPRX1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL19977126 0.81 MRGPRX1 (0.44) MRGPRX1ALDH1A1LMNASMN1; SMN2CYP1A2
SCHEMBL16993907 0.80 MRGPRX1 (0.42) MRGPRX1MAPTALDH1A1MEN1KMT2A
SCHEMBL19977043 0.78 MAPT (0.53) MAPTALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL19976988 0.78 MEN1 (0.52) MRGPRX1MAPTALDH1A1SMN1; SMN2MEN1
SCHEMBL19977073 0.78 PGR (0.52) MAPTF2RALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed