SCHEMBL19981275

SCHEMBL19981275

C[C@H](O)[C@H](NC(=O)N[C@@H](CCC(=O)O)c1nc(-c2cccc(C(F)(F)F)c2)no1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.47
DPP7 Q9UHL4 1/20 0.47
FFAR1 O14842 2/20 0.45
IDH1 O75874 2/20 0.42
VSIR Q9H7M9 2/20 0.42
CD274 Q9NZQ7 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
KCNT1 Q5JUK3 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19981254 0.90 KCNT1 (0.47) FFAR1IDH1VSIRCD274LMNA
SCHEMBL19981256 0.85 VSIR (0.44) FFAR1IDH1VSIRCD274LMNA
SCHEMBL19867036 0.79 VSIR (0.43) DPP4DPP7VSIRCD274LMNA
SCHEMBL18077932 0.79 VSIR (0.43) DPP4DPP7VSIRCD274LMNA
SCHEMBL18077933 0.77 CD274 (0.58) IDH1VSIRCD274LMNATSHR
SCHEMBL19867027 0.77 CD274 (0.58) IDH1VSIRCD274LMNATSHR
SCHEMBL19866982 0.76 VSIR (0.45) VSIRCD274LMNATSHRKCNT1
SCHEMBL18077937 0.76 VSIR (0.45) VSIRCD274LMNATSHRKCNT1
SCHEMBL19962773 0.74 CD274 (0.60) VSIRCD274
SCHEMBL19969881 0.74 CD274 (0.60) VSIRCD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018051254-A1 CYCLIC SUBSTITUTED-1,2,4-OXADIAZOLE COMPOUNDS AS IMMUNOMODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2018-03-22 WO disclosed