SCHEMBL19982254

SCHEMBL19982254

COC(=O)CNC(=O)CC1CCN(C(=O)CCc2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 10/20 0.57
OPRD1 P41143 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
RAB9A P51151 1/20 0.43
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42
PYGL P06737 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
CCR3 P51677 1/20 0.40
DPP4 P27487 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982105 0.84 YAP1 (0.56) YAP1GRIN2B
SCHEMBL19982103 0.82 YAP1 (0.57) YAP1HRH3
SCHEMBL19974601 0.81 YAP1 (0.54) YAP1OPRD1GRIN1GRIN2BCCR3
SCHEMBL21366290 0.80 YAP1 (0.69) YAP1OPRD1
SCHEMBL21366289 0.80 YAP1 (0.69) YAP1OPRD1
SCHEMBL21366352 0.79 YAP1 (0.67) YAP1OPRD1
SCHEMBL21366351 0.79 YAP1 (0.67) YAP1OPRD1
SCHEMBL30117577 0.79 YAP1 (0.79) YAP1
SCHEMBL19982266 0.79 YAP1 (0.79) YAP1
SCHEMBL23339258 0.78 YAP1 (0.69) YAP1OPRD1GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053446-A1 YAP1 INHIBITORS THAT TARGET THE INTERACTION OF YAP1 WITH OCT4 H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2018-03-22 WO disclosed