SCHEMBL19982657

SCHEMBL19982657

CCO[PH](=O)Cc1cccc(COc2ccccc2CC2CCN(Cc3ccc4nc(-c5cccc(C(F)(F)F)c5)[nH]c4c3)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.42
SIGMAR1 Q99720 4/20 0.42
DRD3 P35462 2/20 0.42
TMEM97 Q5BJF2 1/20 0.42
CNR2 P34972 6/20 0.42
CNR1 P21554 1/20 0.42
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
SLC2A1 P11166 1/20 0.39
CHEK2 O96017 4/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19986772 0.94 SLC2A1 (0.42) DRD4SIGMAR1DRD3TMEM97BCHE
SCHEMBL19982671 0.92 BCHE (0.45) BCHEACHECHEK2
SCHEMBL19986769 0.91 DRD4 (0.45) DRD4SIGMAR1DRD3TMEM97CNR2
SCHEMBL19982656 0.88 DRD4 (0.42) DRD4SIGMAR1DRD3TMEM97CNR2
SCHEMBL19970804 0.85 CNR2 (0.40) DRD4SIGMAR1DRD3TMEM97CNR2
SCHEMBL19982651 0.82 CYP1A2 (0.42) DRD4SIGMAR1DRD3TMEM97BCHE
SCHEMBL19982564 0.82 SLC2A1 (0.42) DRD4SIGMAR1DRD3TMEM97BCHE
SCHEMBL19982585 0.80 DRD4 (0.42) DRD4SIGMAR1DRD3TMEM97CNR2
SCHEMBL19982584 0.80 CHEK2 (0.46) BCHEACHECHEK2
SCHEMBL19982583 0.79 SLC2A1 (0.42) DRD4SIGMAR1DRD3TMEM97CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018050771-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-22 WO disclosed
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed