SCHEMBL19982585

SCHEMBL19982585

CCOPCc1cccc(COc2ccccc2CN2CCN(Cc3ccc4nc(-c5cccc(C(F)(F)F)c5)[nH]c4c3)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.42
SIGMAR1 Q99720 4/20 0.42
DRD3 P35462 2/20 0.42
TMEM97 Q5BJF2 1/20 0.42
SLC2A1 P11166 2/20 0.42
CNR2 P34972 7/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
CNR1 P21554 3/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.38
KCNH2 Q12809 1/20 0.37
NPBWR1 P48145 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
XBP1 P17861 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19982583 0.86 SLC2A1 (0.42) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19982612 0.84 CYP1A2 (0.43) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19982610 0.83 SLC2A1 (0.42) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19970766 0.82 SLC2A1 (0.46) SLC2A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL19982656 0.80 DRD4 (0.42) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19982657 0.80 DRD4 (0.42) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19982561 0.80 SLC2A1 (0.46) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19970889 0.78 SLC2A1 (0.44) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19970747 0.78 DRD4 (0.45) DRD4SIGMAR1DRD3TMEM97SLC2A1
SCHEMBL19986769 0.78 DRD4 (0.45) DRD4SIGMAR1DRD3TMEM97SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018050771-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-22 WO disclosed
EP-3296297-A1 BENZIMIDAZOL DERIVATIVES FOR TREATING FILOVIRUS INFECTION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-21 EP disclosed