SCHEMBL19984596

SCHEMBL19984596

CC1=C(C)S(=O)(=O)c2ccc(C(=O)NCc3cnc(-c4ccc(OCCCN(C)C)cc4)s3)cc2NC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.41
ROCK2 O75116 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CHEK2 O96017 1/20 0.37
CHEK1 O14757 2/20 0.36
KDR P35968 2/20 0.36
DAPK3 O43293 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
ABL1 P00519 1/20 0.36
LCK P06239 1/20 0.36
RET P07949 1/20 0.36
MET P08581 1/20 0.36
PDGFRB P09619 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21939692 0.91 ROCK1 (0.42) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21250412 0.88 ROCK1 (0.40) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21939975 0.87 DRD2 (0.41) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21291440 0.86 ROCK1 (0.42) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21250456 0.84 DRD2 (0.39) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21250356 0.83 KMT2A (0.40) DRD2HRH3JAK3ACHEMAPT
SCHEMBL20493939 0.83 MAPT (0.37) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL21250365 0.83 DRD2 (0.37) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL20493937 0.83 MAPT (0.37) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL18667167 0.82 DRD2 (0.36) ROCK1ROCK2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220023311-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES INC (US) 2022-01-27 US disclosed
WO-2018053157-A1 HEPATITIS B CORE PROTEIN MODULATORS ASSEMBLY BIOSCIENCES, INC. (US) 2018-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220023311-A1 HEPATITIS B CORE PROTEIN MODULATORS HAVCR2, FABP1, MAVS ROCK1 4155/4885ROCK2 3592/4885CYP3A4 303/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.