SCHEMBL19986524

SCHEMBL19986524

NC1(CNc2c(Cl)cncc2Cl)CCCC1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.33
BCDIN3D Q7Z5W3 7/20 0.33
MAPT P10636 2/20 0.32
HTT P42858 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
IRAK1 P51617 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28571392 0.80 P2RX7 (0.32) P2RX7
SCHEMBL28576952 0.79 P2RX7 (0.34) P2RX7
SCHEMBL28577549 0.70 CCNT1 (0.30)
SCHEMBL19986728 0.69
SCHEMBL19986641 0.66 STK17A (0.37) P2RX7MAPTHTTCDK5CDK5R1
SCHEMBL28622324 0.65 MAPT (0.31) MAPT
SCHEMBL12212191 0.63 KDM4E (0.37) BCDIN3DIRAK1
SCHEMBL3232274 0.63 MAPK1 (0.41) BCDIN3D
SCHEMBL6221844 0.63 P2RX7 (0.43) P2RX7
Hydrochloric Acid SCHEMBL2518801 0.62 KDM4E (0.36) BCDIN3DIRAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429341-A Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-09-24 CN disclosed
CN-109790123-B Novel capsid protein assembly inhibitors 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed
CN-109790123-A Novel capsid protein assembles inhibitor 正大天晴药业集团股份有限公司 2019-05-21 CN disclosed
WO-2018050110-A1 NOVEL CAPSID PROTEIN ASSEMBLY INHIBITOR 正大天晴药业集团股份有限公司 2018-03-22 WO disclosed