SCHEMBL1999445

SCHEMBL1999445

O=C(c1nc(-c2ccccn2)no1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.41
NPC1 O15118 6/20 0.38
MAPT P10636 5/20 0.38
SMN1; SMN2 Q16637 5/20 0.38
LMNA P02545 4/20 0.38
HTT P42858 2/20 0.38
PPP1CA P62136 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RAB9A P51151 5/20 0.37
TP53 P04637 4/20 0.37
PRCP P42785 1/20 0.36
TSHR P16473 4/20 0.36
MITF O75030 1/20 0.36
PKM P14618 1/20 0.36
EPHX2 P34913 1/20 0.36
AR P10275 1/20 0.36
FAAH O00519 1/20 0.36
CES1 P23141 1/20 0.36
NCEH1 Q6PIU2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005642 0.95 GRM5 (0.39) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL2001115 0.95 GRM5 (0.41) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL2009569 0.95 GRM5 (0.39) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL4564522 0.93 NPC1 (0.38) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL2005062 0.90 EPHX2 (0.33) NPC1MAPTSMN1; SMN2LMNAL3MBTL1
SCHEMBL2011254 0.89 GRM5 (0.45) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL2007450 0.87 LMNA (0.38) GRM5MAPTSMN1; SMN2LMNATP53
SCHEMBL2004941 0.86 GRM5 (0.38) GRM5NPC1MAPTSMN1; SMN2LMNA
SCHEMBL2004659 0.86 KDM4E (0.37) NPC1MAPTLMNAHTTRAB9A
SCHEMBL2003332 0.86 SMN1; SMN2 (0.39) NPC1MAPTSMN1; SMN2LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed