Epinephrine

Epinephrine

SCHEMBL19994728

CNC[C@H](O)c1ccc(O)c(O)c1.Cl.O=[N+]([O-])O

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3

The experimentally established mechanism targets of Epinephrine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 7/20 0.79
ADRB1 known ✓ P08588 5/20 0.77
ADRB3 known ✓ P13945 4/20 0.77
ADRA2A known ✓ P08913 2/20 0.77
ADRA2B known ✓ P18089 2/20 0.77
ADRA2C known ✓ P18825 2/20 0.77
ADRA1D known ✓ P25100 2/20 0.77
ADRA1A known ✓ P35348 2/20 0.77
ADRA1B known ✓ P35368 2/20 0.77
KDM4E B2RXH2 8/20 0.79
BLM P54132 6/20 0.79
PMP22 Q01453 2/20 0.79
NPSR1 Q6W5P4 1/20 0.79
TDP1 Q9NUW8 8/20 0.77
MAPT P10636 7/20 0.77
HSD17B10 Q99714 6/20 0.77
HIF1A Q16665 5/20 0.77
MEN1 O00255 4/20 0.77
KMT2A Q03164 4/20 0.77
TSHR P16473 4/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Racepinephrine SCHEMBL9614373 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Racepinephrine SCHEMBL41370 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Epinephrine SCHEMBL25041 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Racepinephrine SCHEMBL31238229 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Epinephrine SCHEMBL31267207 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Epinephrine SCHEMBL4980185 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
L-Adrenaline SCHEMBL4983607 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Racepinephrine SCHEMBL16667632 0.89 KDM4E (1.00) KDM4EADRB2BLMPMP22NPSR1
Epinephrine SCHEMBL3111795 0.88 KDM4E (0.96) KDM4EADRB2BLMPMP22NPSR1
Racepinephrine SCHEMBL28311143 0.88 KDM4E (0.96) KDM4EADRB2BLMPMP22NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515520-B1 DEVICES AND METHODS FOR VASCULAR HYPERPERFUSION OF EXTRAVASCULAR SPACE ALL VASCULAR PTY LTD (AU) 2024-03-06 EP disclosed
US-20200038575-A1 Devices and Methods for Vascular Hyperperfusion of Extravascular Space All Vascular Pty Limited (AU) 2020-02-06 US disclosed
EP-3515520-A1 DEVICES AND METHODS FOR VASCULAR HYPERPERFUSION OF EXTRAVASCULAR SPACE All Vascular Pty Limited (AU) 2019-07-31 EP disclosed
WO-2018053574-A1 DEVICES AND METHODS FOR VASCULAR HYPERPERFUSION OF EXTRAVASCULAR SPACE All Vascular Pty Limited (AU) 2018-03-29 WO disclosed