SCHEMBL19995580

SCHEMBL19995580

NC(=S)N1CCC[C@@H](c2ccccc2)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
LMNA P02545 2/20 0.50
HPGD P15428 1/20 0.50
HIF1A Q16665 1/20 0.50
DRD2 P14416 1/20 0.50
DRD1 P21728 1/20 0.50
DRD4 P21917 1/20 0.50
DRD5 P21918 1/20 0.50
DRD3 P35462 1/20 0.50
HSD11B1 P28845 2/20 0.49
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
MAPT P10636 2/20 0.48
GAA P10253 1/20 0.48
PARP14 Q460N5 1/20 0.47
PARP10 Q53GL7 1/20 0.47
POLB P06746 2/20 0.47
TSHR P16473 1/20 0.47
RECQL P46063 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19995532 1.00 ALDH1A1 (0.52) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL19995815 0.92 RAB9A (0.56) ALDH1A1LMNAHPGDNPC1RAB9A
SCHEMBL20005696 0.92 RAB9A (0.56) ALDH1A1LMNAHPGDNPC1RAB9A
SCHEMBL19995564 0.92 RAB9A (0.56) ALDH1A1LMNAHPGDNPC1RAB9A
SCHEMBL23009741 0.83 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL27446535 0.83 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL27878990 0.79 ALDH1A1 (0.62) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL3312540 0.79 ALDH1A1 (0.62) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL5230772 0.77 ALDH1A1 (0.43) ALDH1A1LMNAHPGDHIF1ADRD2
SCHEMBL5230779 0.77 ALDH1A1 (0.43) ALDH1A1LMNAHPGDHIF1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515433-A1 BLOOD-BRAIN BARRIER-PENETRANT DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2019-07-31 EP disclosed
WO-2018056854-A1 BLOOD-BRAIN BARRIER-PENETRANT DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2018-03-29 WO disclosed