SCHEMBL20000530

SCHEMBL20000530

c1cc(N2CCCC2)nc(N2CCOCC2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.51
ALDH1A1 P00352 3/20 0.51
PIK3CD O00329 2/20 0.51
MAPK1 P28482 1/20 0.51
PIK3R1 P27986 1/20 0.51
PIK3CB P42338 1/20 0.51
TSHR P16473 2/20 0.50
GBA1 P04062 1/20 0.49
KMT2A Q03164 2/20 0.49
ACHE P22303 2/20 0.48
MEN1 O00255 1/20 0.48
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.48
ALOX15 P16050 1/20 0.48
CYP2C19 P33261 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
OGA O60502 1/20 0.47
ACACB O00763 1/20 0.46
MTOR P42345 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19725018 0.97 PIK3CA (0.49) PIK3CAALDH1A1PIK3CDMAPK1PIK3R1
SCHEMBL5457199 0.95 PIK3CA (0.55) PIK3CAALDH1A1PIK3CDPIK3R1PIK3CB
SCHEMBL8549105 0.89 GBA1 (0.56) GBA1ACHESORDCCNT1CCNA2
SCHEMBL27941842 0.88 GBA1 (0.55) GBA1ACHESORDCCNT1CCNA2
SCHEMBL30635502 0.88 GBA1 (0.55) GBA1ACHESORDCCNT1CCNA2
SCHEMBL30818658 0.87 HRH3 (0.51) PIK3CAALDH1A1PIK3CDPIK3R1PIK3CB
SCHEMBL1123812 0.84 MAPT (0.58) PIK3CAALDH1A1PIK3CDPIK3R1PIK3CB
SCHEMBL5485306 0.83 PIK3CA (0.49) PIK3CAALDH1A1PIK3CDPIK3R1PIK3CB
SCHEMBL28637136 0.80 CASP1 (0.67) ALDH1A1GBA1ACHEUSP2CYP1A2
SCHEMBL29519526 0.80 CASP1 (0.67) ALDH1A1GBA1ACHEUSP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997024-B1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2018-03-28 EP disclosed