SCHEMBL20001656

SCHEMBL20001656

CN(C)CCNc1ccc(C(=N)N)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 9/20 0.66
F2 P00734 3/20 0.64
PRSS2 P07478 3/20 0.64
PRSS3 P35030 3/20 0.64
TMPRSS6 Q8IU80 3/20 0.64
ST14 Q9Y5Y6 3/20 0.64
KLK1 P06870 1/20 0.46
KLK5 Q9Y337 1/20 0.46
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAOA P21397 1/20 0.43
CNR1 P21554 1/20 0.43
DRD4 P21917 1/20 0.43
ACHE P22303 1/20 0.43
HRH2 P25021 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3872851 0.85 PRSS1 (0.60) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL3875680 0.83 PRSS1 (0.84) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL3667557 0.80 PRSS1 (0.72) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL3869914 0.80 PRSS1 (0.57) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL5524345 0.80 PRSS1 (1.00) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL17515720 0.78 PRSS1 (0.75) PRSS1F2PRSS2PRSS3TMPRSS6
SCHEMBL4135587 0.77 LMNA (0.51) LMNACYP1A2MAOACNR1DRD4
SCHEMBL3689477 0.77 LMNA (0.51) LMNACYP1A2MAOACNR1DRD4
Hydrochloric Acid SCHEMBL5071263 0.76 LMNA (0.52) LMNACYP1A2MAOACNR1DRD4
SCHEMBL6318640 0.76 HRH3 (0.46) LMNACYP1A2MAOACNR1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018054989-A1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2018-03-29 WO disclosed