SCHEMBL2000292

SCHEMBL2000292

O=C(c1nc(-c2ccncc2)no1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.41
SMPD1 P17405 3/20 0.38
TSHR P16473 2/20 0.37
GSK3B P49841 1/20 0.37
CNR2 P34972 1/20 0.37
STAT3 P40763 1/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
TP53 P04637 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
MAPT P10636 3/20 0.36
HDAC8 Q9BY41 2/20 0.36
RAB9A P51151 1/20 0.36
DUSP3 P51452 1/20 0.36
PTPN11 Q06124 1/20 0.36
LMNA P02545 1/20 0.36
THRB P10828 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002246 0.94 SMN1; SMN2 (0.39) SMN1; SMN2SMPD1CNR2STAT3HDAC1
SCHEMBL2004417 0.93 TP53 (0.44) SMN1; SMN2SMPD1CNR2STAT3HDAC1
SCHEMBL2005271 0.92 TSHR (0.43) SMN1; SMN2SMPD1TSHRTP53MAPT
SCHEMBL2002094 0.91 SMN1; SMN2 (0.43) SMN1; SMN2SMPD1TSHRGSK3BCNR2
SCHEMBL2003332 0.91 SMN1; SMN2 (0.39) SMN1; SMN2TSHRGSK3BCNR2HDAC6
SCHEMBL2000479 0.90 CYP1A2 (0.44) SMN1; SMN2TSHRGSK3BCNR2HDAC1
SCHEMBL2001517 0.90 ALOX5AP (0.42) SMN1; SMN2SMPD1TSHRCNR2STAT3
SCHEMBL2002063 0.88 ALOX5 (0.33) SMN1; SMN2SMPD1TSHRSTAT3MAPT
SCHEMBL2004345 0.88 SMPD1 (0.41) SMN1; SMN2SMPD1TSHRGSK3BTP53
SCHEMBL2002547 0.86 RAB9A (0.39) SMN1; SMN2TSHRGSK3BCNR2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed