SCHEMBL20002979

SCHEMBL20002979

COc1cc(C#N)ccc1COC(C)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.47
NR3C1 P04150 7/20 0.44
NR3C2 P08235 7/20 0.44
PGR P06401 6/20 0.44
AR P10275 3/20 0.40
PTGES2 Q9H7Z7 2/20 0.38
CETP P11597 2/20 0.38
SLC6A4 P31645 1/20 0.36
CFB P00751 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19387995 0.85 AR (0.43) RORCNR3C1NR3C2PGRAR
SCHEMBL20002764 0.83 NR3C1 (0.46) RORCNR3C1NR3C2PGRCETP
SCHEMBL16892231 0.79 AR (0.47) RORCNR3C1NR3C2PGRAR
SCHEMBL1715169 0.76 IDO1 (0.51) RORCARPTGES2SLC6A4
Hydrochloric Acid SCHEMBL1715038 0.75 IDO1 (0.53) RORCARPTGES2SLC6A4
SCHEMBL1855982 0.74 AR (0.49) ARPTGES2SLC6A4TRPV4
SCHEMBL7667004 0.72 AR (0.47) NR3C1NR3C2PGRARPTGES2
SCHEMBL3288455 0.72 AR (0.47) ARPTGES2SLC6A4
SCHEMBL22481567 0.72 AR (0.47) NR3C1NR3C2PGRARPTGES2
SCHEMBL3571001 0.72 AR (0.47) PGRARCFBTRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed