SCHEMBL20002764

SCHEMBL20002764

CC(OCc1ccc(C#N)cc1F)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.46
PGR P06401 2/20 0.46
NR3C2 P08235 2/20 0.46
RORC P51449 4/20 0.44
CETP P11597 2/20 0.39
KIF11 P52732 1/20 0.38
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
KCNH2 Q12809 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
IDO1 P14902 1/20 0.35
MAPK14 Q16539 1/20 0.34
SLC22A12 Q96S37 1/20 0.34
CTSB P07858 1/20 0.34
PRMT5 O14744 1/20 0.34
EGFR P00533 1/20 0.34
TRPV4 Q9HBA0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19387997 0.86 NR3C1 (0.43) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL20002979 0.83 RORC (0.47) NR3C1PGRNR3C2RORCCETP
SCHEMBL20002813 0.80 IDO1 (0.53) NR3C1PGRNR3C2RORCIDO1
SCHEMBL3641589 0.78 NR3C1 (0.43) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL29506809 0.78 NR3C1 (0.43) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL23286946 0.75 FFAR1 (0.41) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL1715728 0.74 IDO1 (0.59) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL13315163 0.74 NR3C1 (0.48) NR3C1PGRNR3C2KIF11FFAR1
SCHEMBL21086643 0.74 FFAR1 (0.39) NR3C1PGRNR3C2RORCFFAR1
SCHEMBL16841663 0.74 FFAR1 (0.40) NR3C1PGRNR3C2RORCCETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed