SCHEMBL20004149

SCHEMBL20004149

COc1cc2c(cc1[S+]([O-])N1CCN(C)CC1)Cc1c([nH]c3cc(Br)ccc13)C2(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 15/20 0.50
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR1A P08908 1/20 0.30
CYP2D6 P10635 1/20 0.30
DRD2 P14416 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21443150 0.82 ALK (0.35) ALKHTR6
SCHEMBL20004151 0.81 ALK (0.51) ALKCA1CA2CA4CA6
SCHEMBL17448483 0.81 ALK (0.43) ALK
SCHEMBL897744 0.80 ALK (0.50) ALKCA1CA2CA4CA6
SCHEMBL897370 0.79 ALK (0.75) ALK
SCHEMBL16775676 0.79 ALK (0.47) ALKCA1CA2CA4CA6
SCHEMBL27087539 0.78 ALK (0.48) ALKCA1CA2CA4CA6
SCHEMBL7806147 0.78 ALK (0.63) ALKCYP1A2CYP3A4HTR1ACYP2D6
SCHEMBL20366555 0.77 ALK (0.31) ALK
SCHEMBL27087566 0.77 ALK (0.47) ALKCA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed