SCHEMBL20004502

SCHEMBL20004502

Cc1ccc(COCc2ccncc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.52
AGXT P21549 2/20 0.50
NPC1 O15118 2/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 4/20 0.43
RAB9A P51151 2/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
MMP13 P45452 2/20 0.41
MMP2 P08253 1/20 0.41
CYP3A4 P08684 1/20 0.41
STAT3 P40763 1/20 0.41
MAPK14 Q16539 1/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3161372 0.86 AGXT (0.64) KCNH2AGXTNPC1SMN1; SMN2RAB9A
SCHEMBL9617939 0.86 AGXT (0.64) KCNH2AGXTNPC1SMN1; SMN2RAB9A
SCHEMBL492258 0.86 TSHR (0.52) KMT2ALMNAALDH1A1TSHRCYP3A4
Lithium SCHEMBL585057 0.84 AGXT (0.61) KCNH2AGXTNPC1SMN1; SMN2RAB9A
Potassium SCHEMBL586332 0.84 AGXT (0.61) KCNH2AGXTNPC1SMN1; SMN2RAB9A
SCHEMBL586154 0.84 AGXT (0.61) KCNH2AGXTNPC1SMN1; SMN2RAB9A
Hydrochloric Acid SCHEMBL27794104 0.84 TSHR (0.50) KMT2ALMNAALDH1A1TSHRCYP3A4
SCHEMBL22537715 0.83 RAB9A (0.46) KCNH2NPC1KMT2ASMN1; SMN2RAB9A
SCHEMBL8361590 0.79 NPC1 (0.58) KCNH2NPC1KMT2ASMN1; SMN2RAB9A
SCHEMBL171160 0.79 CYP17A1 (0.54) NPC1KMT2ASMN1; SMN2RAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515912-B1 COMPOUNDS FOR USING IN IMAGING AND PARTICULARLY FOR THE DIAGNOSIS OF NEURODEGENERATIVE DISEASES CENTRE NAT RECH SCIENT (FR) 2020-10-14 EP disclosed
WO-2018055316-A1 COMPOUNDS FOR USING IN IMAGING AND PARTICULARLY FOR THE DIAGNOSIS OF NEURODEGENERATIVE DISEASES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2018-03-29 WO disclosed