SCHEMBL20005289

SCHEMBL20005289

Cc1ccc(-c2ccc(-c3cc(C)c(C#Cc4cc(F)c(F)c(F)c4)c(F)c3)c(F)c2)c(F)c1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.33
AKR1C2 P52895 2/20 0.33
PDE3B Q13370 5/20 0.32
PDE3A Q14432 5/20 0.32
AKR1B10 O60218 1/20 0.32
AKR1C4 P17516 1/20 0.32
AKR1C1 Q04828 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20004795 0.96 GRM5 (0.34) AKR1C3AKR1C2PDE3BPDE3AAKR1B10
SCHEMBL20004915 0.95 PDE3B (0.33) AKR1C3AKR1C2PDE3BPDE3A
SCHEMBL20005288 0.94 PDE3B (0.32) AKR1C3AKR1C2PDE3BPDE3AAKR1B10
SCHEMBL20005243 0.92 PDE9A (0.33) PDE3BPDE3A
SCHEMBL20004646 0.91 KDM1A (0.31) PDE3BPDE3A
SCHEMBL20004910 0.90 GRM5 (0.33) AKR1C3AKR1C2PDE3BPDE3AAKR1B10
SCHEMBL19999441 0.90 GRM5 (0.34) AKR1C3AKR1C2PDE3BPDE3AAKR1B10
SCHEMBL20005252 0.89 PDE3B (0.33) PDE3BPDE3A
SCHEMBL20005223 0.88 GRM5 (0.34) PDE3BPDE3AGRM5
SCHEMBL20006757 0.88 TNKS (0.40) AKR1C3AKR1C2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299439-A1 LIQUID CRYSTAL COMPOUND, LIQUID CRYSTAL COMPOSITION AND LIQUID CRYSTAL DISPLAY DEVICE JNC Corporation (JP) 2018-03-28 EP disclosed